AG 1433 HCl分子式: C16H14N2O2·HCl分子量: 302.76描述应用储存/保存方法形态别名沸点折射率IC50可溶性/溶解性MDL
产品描述 | |
描述 |
AG 1433 Hydrochloride is a specific and potent inhibitor of platelet-derived growth factor-β receptor kinase (PDGF-β receptor kinase, IC50 = 5.0 μM) and of Flk-1/KDR/VEGF Receptor 2 (IC50 = 9.3 μM). AG 1433 Hydrochloride also acts as angiogenesis inhibitor.
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应用 |
A PDGF-β receptor kinase and angiogenesis inhibitor
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储存/保存方法 |
Store at -20° C
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形态 |
Solid
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基本信息 | |
别名 |
2-(3,4-Dihydroxyphenyl)-6,7-dimethylquinoxaline
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沸点 |
511.7° C at 760 mmHg (Predicted)
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折射率 |
n20D ~1.69 (Predicted)
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IC50 |
PDGFR-beta: IC50 = 5 µM; Flk-1: IC50 = 9.3 µM
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可溶性/溶解性 |
DMSO (3 mg/ml). Further dilute with aqueous buffers just before use.
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MDL |
MFCD03490489
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