Philanthotoxin 74CAS号： 401601-12-5分子式： C24H42N4O3 2HCl分子量： 507.54描述应用纯度储存/保存方法形态折射率光学活性IC50Ki 数据可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
Subtype-selective AMPA receptor antagonist that inhibits GluR1/2 but not GluR2/3 receptors.
|
| 应用 |
An AMPA receptor antagonist
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| 纯度 |
≥98%
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| 储存/保存方法 |
Desiccate at room temperature
|
| 形态 |
Solid
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| 基本信息 | |
| 折射率 |
n20D 1.53 (Predicted)
|
| 光学活性 |
α20/D +1°, c = 2 in water
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| IC50 |
Glutamate receptor ionotropic, AMPA: IC50 = 138 nM (rat)
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| Ki 数据 |
GluR-1: Ki= 168 nM (human); Glutamate receptor ionotropic, AMPA 1: Ki= 168 nM (rat)
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| 可溶性/溶解性 |
Soluble in water (100 mM), and DMSO (100 mM).
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| MDL |
MFCD09971136
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| PubChem CID |
46213501
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