PF-06821497CAS号： 1844849-10-0分子式： C22H24Cl2N2O5分子量： 467.34描述纯度储存/保存方法可溶性/溶解性靶点In vivo(体内研究)
| 产品描述 | |
| 描述 |
PF-06821497 is a selective inhibitor of EZH2 with significant tumor growth inhibition.
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| 纯度 |
98%
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| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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| 基本信息 | |
| 可溶性/溶解性 |
DMSO:55 mg/mL (117.69 mM)
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| 生物活性 | |
| 靶点 |
Y641N EZH2(ki):ki:<0.1 nM
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| In vivo(体内研究) |
The tumor regression effect of PF-06821497 can be sustained for another 40 days[1].
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