ELN-441958CAS号： 913064-47-8分子式： C29H29ClN4O2分子量： 501.02描述纯度储存/保存方法可溶性/溶解性靶点
| 产品描述 | |
| 描述 |
ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM. ELN-441958 is highly selective for B1 over B2 receptors, and >500/ 2000-fold selective for the B1 over _mu_/_delta_-opioid receptor. |
| 纯度 |
≥98%
|
| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
|
| 基本信息 | |
| 可溶性/溶解性 |
DMSO : 100 mg/mL (199.59 mM; Need ultrasonic)
|
| 生物活性 | |
| 靶点 |
Bradykinin Receptor
|
分子结构图
