CP 376395 hydrochloride

CP 376395 hydrochlorideCAS号: 175140-00-8分子式: C21H30N2•HCl分子量: 362.94描述应用储存/保存方法形态别名折射率IC50Ki 数据可溶性/溶解性MDLPubChem CID

产品描述
描述
CP 376395 hydrochloride is a CRF-RI receptor antagonist which is potent and selective (Ki values are 12 and >10000 nM for CRF-RI and CRF-RII receptors respectively).
应用
A CRF-RI receptor antagonist
储存/保存方法
Store at room temperature
形态
Solid
基本信息
别名
N-(1-Ethylpropyl)-3,6-dimethyl-2-(2,4,6-trimethylphenoxy)-4-pyridinamine hydrochloride
折射率
n20D 1.56 (Predicted)
IC50
Corticotropin releasing factor receptor 1: IC50 = 5.1 nM (rat)
Ki 数据
CRF1 receptor: Ki= 12 nM; CRF2 receptor: Ki= >10 µM
可溶性/溶解性
Soluble in water (50 mM), and DMSO (100 mM).
MDL
MFCD11519966
PubChem CID
24806455