A-437203CAS号： 220519-06-2分子式： C20H27F3N6OS分子量： 456.53描述纯度储存/保存方法别名可溶性/溶解性靶点In vitro(体外研究)In vivo(体内研究)
| 产品描述 | |
| 描述 |
A-437203 is a selective D3 receptor antagonist with Ki of 71, 1.6, and 6220 nM for D2, D3, and D4 receptors, respectively.
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| 纯度 |
98%
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| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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| 基本信息 | |
| 别名 |
ABT-925；A37203； Lu201640
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| 可溶性/溶解性 |
DMSO*
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| 生物活性 | |
| 靶点 |
D2 receptor,D3 receptor,D4 receptor
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| In vitro(体外研究) |
A-437203 is an antagonist with high affinity for D3 receptors and relatively high selectivity compared to other dopamine receptor subtypes (44-fold selective for D3 vs D2).
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| In vivo(体内研究) |
A-437203 is an antagonist with high affinity for D3 receptors and relatively high selectivity compared to other dopamine receptor subtypes (44-fold selective for D3 vs D2).
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分子结构图
