L-368,899 hydrochlorideCAS号： 148927-60-0分子式： C26H42N4O5S2•HCl分子量： 591.22描述应用纯度储存/保存方法形态沸点折射率光学活性IC50可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
L-368,899 hydrochloride is a potent, non-peptide Oxytocin Receptor Inhibitor. L-368,899 hydrochloride has shown a 40-fold selectivity over AVP Receptor V1a (vasopressin V1a) and V2 receptors. L-368,899 hydrochloride has also been shown to antagonize oxytocin-induced uterine contractions in vitro.
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| 应用 |
A non-peptide Oxytocin Receptor Inhibitor
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| 纯度 |
>97%
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| 储存/保存方法 |
Store at -20° C
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| 形态 |
Solid
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| 基本信息 | |
| 沸点 |
794.1° C at 760 mmHg (Predicted)
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| 折射率 |
n20D 1.61 (Predicted)
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| 光学活性 |
α20/D +27°, c = 1 in methanol
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| IC50 |
Oxytocin receptor: IC50 = 8.9 nM; AVP Receptor V1a: IC50 = 370 nM; AVP Receptor V2: IC50 = 570 nM
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| 可溶性/溶解性 |
Soluble in water (100 mM), and DMSO (100 mM).
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| MDL |
MFCD09753328
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| PubChem CID |
56972193
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