SR 3677 hydrochlorideCAS号: 1072959-67-1 (free base)分子式: C22H24N4O4•2HCl分子量: 481.37描述纯度储存/保存方法形态别名外观IC50可溶性/溶解性
产品描述 | |
描述 |
SR 3677 dihydrochloride is a selective and potent Rho-kinase inhibitor IC50 = 3 and 56 nM for ROCK2 and ROCK1, respectively). |
纯度 |
≥98%
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储存/保存方法 |
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
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形态 |
Solid
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基本信息 | |
别名 |
SR 3677 2HCl
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外观 |
Powder
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IC50 |
Rock-2: IC50 = 3 nM; Rock-1: IC50 = 56 nM; Akt: IC50 = 7.49 µM (human)
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可溶性/溶解性 |
Soluble in water (100 mM), and DMSO (100 mM).
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分子结构图