GGTI-298CAS号： 180977-44-0分子式： C27H33N3O3S•CF3CO2H分子量： 593.66描述应用纯度储存/保存方法形态熔点沸点IC50可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
GGTI 298 has been shown to be a CAAZ peptidomimetic GGTase I (geranylgeranyltransferase I) inhibitor. This compound has been shown to cause G0-G1 cell cycle block and apoptosis in A549 cells.
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| 应用 |
A CAAZ peptidomimetic GGTase I inhibitor
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| 纯度 |
≥95%
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| 储存/保存方法 |
Store at -20° C
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| 形态 |
Solid
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| 基本信息 | |
| 熔点 |
99.5-100° C
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| 沸点 |
734.1° C at 760 mmHg (Predicted)
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| IC50 |
Inhibits the processing of geranylgeranylated Rap1A: IC50 = 3 µM; Inhibits the processing of farnesylated Ha-Ras: IC50 >10 µM
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| 可溶性/溶解性 |
Soluble in DMSO (25 mM).
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| MDL |
MFCD06409252
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| PubChem CID |
16078971
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