BML-267分子式： C11H12N2O5S•C2HF3O2分子量： 398.31描述应用纯度储存/保存方法形态别名IC50可溶性/溶解性
| 产品描述 | |
| 描述 |
BML-267 is a potent and selective PTP1B (protein tyrosine phosphatase 1B) inhibitor (IC50=11 μM)1. A similar N-des-methyl analog has been reported and has been used to probe the mechanism of PTP1B-mediated inhibition of leptin signaling. BML-267 have limited cell permeability. A cell permeable diethyl ester prodrug of BML-267 compound is available.
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| 应用 |
A potent and selective protein tyrosine phosphatase 1B (PTP1B) inhibitor
|
| 纯度 |
≥95%
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| 储存/保存方法 |
Store at -20° C
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| 形态 |
Solid
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| 基本信息 | |
| 别名 |
6-Methyl-2-(oxalylamino)-4,5,6,7-tetrahydrothieno[2, 3-c]pyridine-3-carboxylic acid trifluoroacetic acid salt
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| IC50 |
protein tyrosine phosphatase 1B (PTP1B): IC50 = 11 µM
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| 可溶性/溶解性 |
Soluble in: DMSO 10 mg/mL
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