GX 201CAS号： 1788071-27-1分子式： C25H27ClF4N2O4S分子量： 563描述纯度储存/保存方法可溶性/溶解性In vivo(体内研究)
| 产品描述 | |
| 描述 |
GX 201 is a selective NaV1.7 inhibitor, IC50 of < 3.2 nM for hNaV1.7.
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| 纯度 |
98%
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| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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| 基本信息 | |
| 可溶性/溶解性 |
DMSO:60 mg/mL (106.6 mM)
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| 生物活性 | |
| In vivo(体内研究) |
GX 201 has a relatively long half-life in mice. GX 201 produces analgesia at a free plasma concentration about 3 times the IC50 for high-affinity channel block. GX 201 inhibits nociceptive responses induced by formalin and inflammatory pain caused by complete Freund’s adjuvant (CFA)[1].
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