AR-R17779 HClCAS号： 178419-47-1分子式： C9H14N2O2·HCl分子量： 218.68描述应用纯度储存/保存方法形态外观沸点折射率光学活性IC50Ki 数据可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
AR-R17779 HCl is a selective agonist of α7 AChRs (Ki values are 190 and 16000 nM for rat α7 and α4β2 receptors, respectively).
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| 应用 |
A selective agonist of α7 AChRs
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| 纯度 |
≥99%
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| 储存/保存方法 |
Store at room temperature
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| 形态 |
Solid
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| 基本信息 | |
| 外观 |
Powder
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| 沸点 |
411.7° C at 760 mmHg (Predicted)
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| 折射率 |
n20D 1.59 (Predicted)
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| 光学活性 |
α20/D -62.7°, c = 1 in methanol
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| IC50 |
AChRα7: EC5050 = 420 nM (human); Neuronal acetylcholine receptor protein alpha-7 subunit: EC5050 = 21 µM (rat)
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| Ki 数据 |
AChRα7: Ki= 92 nM (human); α7 receptor : Ki= 190 nM (rat); α4β2 receptors : Ki= 16 µM (rat)
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| 可溶性/溶解性 |
Soluble in DMSO (50 mM).
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| MDL |
MFCD20926337
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| PubChem CID |
5310971
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