A 841720CAS号： 869802-58-4分子式： C17H21N5OS分子量： 343.45描述应用纯度储存/保存方法形态可溶性/溶解性PubChem CID
| 产品描述 | |
| 描述 |
A 841720 is a potent, non-competitive mGluR-1 antagonist that displays 34-fold selectivity over mGluR-5 (IC50 values are 10 and 342 nM respectively). A 841720 displays no significant activity at a range of other GPCRs, ion channels and transporters. This compound also exhibits analgesic effects, decreases mechanical allodynia in models of neuropathic pain, and impairs cognitive function.
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| 应用 |
A potent & non-competitive mGluR-1 antagonist
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| 纯度 |
≥98%
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| 储存/保存方法 |
Store at room temperature
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| 形态 |
Solid
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| 基本信息 | |
| 可溶性/溶解性 |
Soluble to 50 mM in DMSO and to 50 mM in Ethanol
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| PubChem CID |
11559235
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