BucolomeCAS号: 841-73-6分子式: C14H22N2O3分子量: 266.34描述纯度储存/保存方法可溶性/溶解性In vitro(体外研究)
产品描述 | |
描述 |
Bucolome is a CYP2C9 inhibitor with uricosuric and anti-inflammatory activity.
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纯度 |
98%
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储存/保存方法 |
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
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基本信息 | |
可溶性/溶解性 |
DMSO:50 mg/mL (187.73 mM)
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生物活性 | |
In vitro(体外研究) |
In studies with recombinant human cytochrome P-450 2C9 and liver microsomes, Bucolome is a potent mixed-type inhibitor for (S)-warfarin 7-hydroxylation, with Ki of 8.2 and 20.2 microM, respectively[1].
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