Bucolome

BucolomeCAS号: 841-73-6分子式: C14H22N2O3分子量: 266.34描述纯度储存/保存方法可溶性/溶解性In vitro(体外研究)

产品描述
描述
Bucolome is a CYP2C9 inhibitor with uricosuric and anti-inflammatory activity.
纯度
98%
储存/保存方法
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
基本信息
可溶性/溶解性
DMSO:50 mg/mL (187.73 mM)
生物活性
In vitro(体外研究)
In studies with recombinant human cytochrome P-450 2C9 and liver microsomes, Bucolome is a potent mixed-type inhibitor for (S)-warfarin 7-hydroxylation, with Ki of 8.2 and 20.2 microM, respectively[1].