L-803,087 trifluoroacetateCAS号： 217480-26-7分子式： C25H29F2N5O3•CF3CO2H分子量： 599.56描述应用纯度储存/保存方法形态别名沸点折射率Ki 数据可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
Potent and selective sst4 agonist Potent and selective somatostatin sst4 receptor agonist. Ki values are 0.7, 199, 4720, 1280 and 3880 nM for cloned human sst4, sst1, sst2, sst3 and sst5 receptors respectively. Facilitates AMPA-mediated hippocampal synaptic responses in vitro.
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| 应用 |
A potent and selective sst4 agonist
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| 纯度 |
≥97%
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| 储存/保存方法 |
Store at -20° C
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| 形态 |
Solid
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| 基本信息 | |
| 别名 |
N2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-arginine methyl ester trifluoroacetate; Methyl N2-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)butanoyl]-L-argininate trifluoroacetate;
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| 沸点 |
779.7° C at 760 mmHg (Predicted)
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| 折射率 |
n20D 1.61 (Predicted)
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| Ki 数据 |
SSTR4: Ki= 0.7 nM (human); SSTR1: Ki= 199 nM (human); SSTR3: Ki= 1.28 µM (human); SSTR5: Ki= 3.88 µM (human); SSTR2: Ki= 4.72 µM (human)
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| 可溶性/溶解性 |
Soluble in DMSO (100 mM), and ethanol (100 mM).
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| MDL |
MFCD09037334
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| PubChem CID |
45073436
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