MT-802CAS号： 2231744-29-7分子式： C41H41N9O8分子量： 787.82描述纯度储存/保存方法可溶性/溶解性靶点In vitro(体外研究)
| 产品描述 | |
| 描述 |
MT-802 is an effective BTK degrader based on PROTAC technology (DC50: 1 nM). MT-802 has the potential to treat C481S mutant chronic lymphocytic leukemia (CLL).
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| 纯度 |
97%
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| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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| 基本信息 | |
| 可溶性/溶解性 |
DMSO:100 mg/mL (126.93 mM)
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| 生物活性 | |
| 靶点 |
BTK:1 nM(DC50)
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| In vitro(体外研究) |
MT-802 degrades BTK (DC50: 9.1 nM). The maximal degradation was observed by 250 nM.
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