L-798106CAS号： 244101-02-8分子式： C27H22BrNO4S分子量： 536.44描述应用纯度储存/保存方法形态密度折射率PK值Ki 数据可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
L-798,106 is a potent and highly selective prostanoid EP3 receptor antagonist (Ki values are 0.3, 916, > 5000 and > 5000 nM at EP3, EP4, EP1 and EP2, respectively). Attenuates sulprostone-induced inhibition of EFS-evoked twitch and contractile responses in vivo.
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| 应用 |
A potent and highly selective prostanoid EP3 receptor antagonist
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| 纯度 |
≥98%
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| 储存/保存方法 |
Store at 4° C
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| 形态 |
Solid
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| 基本信息 | |
| 密度 |
1.43 g/cm3 (Predicted)
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| 折射率 |
n20D 1.66 (Predicted)
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| PK值 |
pKa: 4.26 (Predicted)
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| Ki 数据 |
EP3: Ki= 0.3 nM; IP Receptor: Ki= >500 nM (human); PGF2Rα receptor: Ki= >500 nM (human); DP: Ki= >500 nM (human); TXA2R: Ki= >500 nM (human)
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| 可溶性/溶解性 |
Soluble in DMSO (100 mM).
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| MDL |
MFCD08272644
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| PubChem CID |
15551229
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