MG 624CAS号： 77257-42-2分子式： C22H30NOI分子量： 451.39描述应用储存/保存方法形态熔点IC50Ki 数据可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
MG 624 is a neuronal AChR α7 antagonist. MG 624 inhibits α-Bgtx binding to chick α7 and α4β2 subtypes.
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| 应用 |
An antagonist of neuronal AChR
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| 储存/保存方法 |
Desiccate at 4° C
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| 形态 |
Solid
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| 基本信息 | |
| 熔点 |
212-213° C
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| IC50 |
Plasmodium falciparum: IC50 = 0.40 µM; APOBEC503A: IC50 = 2.33 µM (human); APOBEC503G: IC50 = 2.57 µM (human); CTDSP1: IC50 = 20.22 µM (human)
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| Ki 数据 |
Inhibits α-Bgtx binding to chick α7 and α4β2 subtypes with Kivalues of 106 nM and 84 µM respectively
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| 可溶性/溶解性 |
Soluble in DMSO (20 mM), and ethanol (10 mM). Insoluble in water.
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| MDL |
MFCD00865233
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| PubChem CID |
6433339
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