GSK3326595

GSK3326595 CAS号: 1616392-22-3分子式: C24H32N6O3分子量: 452.55描述纯度储存/保存方法别名外观可溶性/溶解性靶点In vitro(体外研究)

产品描述
描述
GSK3326595 (EPZ015938) is a potent, selective, reversible inhibitor of protein arginine methyltransferase 5 (PRMT5) with an IC50 of 6.2 nM.
纯度
≥98%
储存/保存方法
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
基本信息
别名
EPZ015938;GSK-3326595
外观
Off-white solid
可溶性/溶解性
DMSO : 66.67 mg/mL (147.32 mM; Need ultrasonic)
生物活性
靶点
Histone Methyltransferase
In vitro(体外研究)
GSK3326595 (EPZ015938), has entered clinical trials for the treatment of solid tumors and non-Hodgkin’s lymphoma.

分子结构图

GSK3326595