GSK3326595 CAS号: 1616392-22-3分子式: C24H32N6O3分子量: 452.55描述纯度储存/保存方法别名外观可溶性/溶解性靶点In vitro(体外研究)
产品描述 | |
描述 |
GSK3326595 (EPZ015938) is a potent, selective, reversible inhibitor of protein arginine methyltransferase 5 (PRMT5) with an IC50 of 6.2 nM.
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纯度 |
≥98%
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储存/保存方法 |
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
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基本信息 | |
别名 |
EPZ015938;GSK-3326595
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外观 |
Off-white solid
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可溶性/溶解性 |
DMSO : 66.67 mg/mL (147.32 mM; Need ultrasonic)
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生物活性 | |
靶点 |
Histone Methyltransferase
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In vitro(体外研究) |
GSK3326595 (EPZ015938), has entered clinical trials for the treatment of solid tumors and non-Hodgkin’s lymphoma.
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分子结构图