NNC 63-0532CAS号： 250685-44-0分子式： C27H29N3O3分子量： 443.54描述应用储存/保存方法形态密度熔点沸点折射率IC50PK值Ki 数据可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
NNC 63-0532 is a potent non-peptide agonist for the KOR-3 (NOP receptor) (EC50 = 305 nM, Ki = 7.3 nM); about a 12-fold increase in selectivity over other receptors.
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| 应用 |
A potent non-peptide agonist for the NOP receptor
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| 储存/保存方法 |
Store at room temperature
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| 形态 |
Solid
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| 基本信息 | |
| 密度 |
~1.3 g/cm3 (Predicted)
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| 熔点 |
259.06° C (Predicted)
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| 沸点 |
~645.8° C at 760 mmHg (Predicted)
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| 折射率 |
n20D 1.68 (Predicted)
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| IC50 |
NOP receptor: EC5050 = 305 nM
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| PK值 |
pKb: 8.39 (Predicted)
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| Ki 数据 |
NOP receptor: Ki= 7.3 nM
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| 可溶性/溶解性 |
Soluble in ethanol (5 mM), and DMSO (50 mM).
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| MDL |
MFCD04113779
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| PubChem CID |
9803475
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