PF 05089771

PF 05089771CAS号: 1235403-62-9分子式: C18H12Cl2FN5O3S2分子量: 500.35描述纯度储存/保存方法外观可溶性/溶解性靶点

产品描述
描述
PF 05089771 is a potent, orally active and selective arylsulfonamide Nav1.7 inhibitor, with IC50 values of 11 nM, 12 nM, 13 nM, 171 nM and 8 nM for hNav1.7, cynNav1.7, dogNav1.7, ratNav1.7, and musNav1.7, respectively. PF 05089771 is under the study for pain and diabetic neuropathy.
纯度
98%
储存/保存方法
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
基本信息
外观
White solid
可溶性/溶解性
DMSO : 100 mg/mL (199.86 mM; Need ultrasonic)
生物活性
靶点
Sodium Channel

分子结构图

PF 05089771