PF 05089771CAS号: 1235403-62-9分子式: C18H12Cl2FN5O3S2分子量: 500.35描述纯度储存/保存方法外观可溶性/溶解性靶点
产品描述 | |
描述 |
PF 05089771 is a potent, orally active and selective arylsulfonamide Nav1.7 inhibitor, with IC50 values of 11 nM, 12 nM, 13 nM, 171 nM and 8 nM for hNav1.7, cynNav1.7, dogNav1.7, ratNav1.7, and musNav1.7, respectively. PF 05089771 is under the study for pain and diabetic neuropathy.
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纯度 |
98%
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储存/保存方法 |
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
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基本信息 | |
外观 |
White solid
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可溶性/溶解性 |
DMSO : 100 mg/mL (199.86 mM; Need ultrasonic)
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生物活性 | |
靶点 |
Sodium Channel
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分子结构图