PNU 96415E

PNU 96415ECAS号: 170856-41-4分子式: C21H25FN2O•2HCl分子量: 413.36描述应用纯度储存/保存方法形态别名可溶性/溶解性

产品描述
描述
PNU 96415E is chemically unrelated to clozapine, an antipsychotic agent. PNU 96415E displays highest affinity for dopamine D4 and SR-2A and relatively weak affinity at D2 receptors (Ki values are 3.0, 5.8, 134, 181, 199, 240, 411 and > 678 nM for D4, SR-2A, SR-1A, α1, D2, D3, D1, α2 and muscarinic receptors respectively).
应用
A SR-2A inhibitor
纯度
≥98%
储存/保存方法
Desiccate at room temperature
形态
Solid
基本信息
别名
1-[2-(3,4-dihydro-1H-2-benzopyran-1-yl)ethyl]-4-(4-fluorophenyl)piperazine dihydrochloride
可溶性/溶解性
Soluble to 10 mM in Water