CPI-637CAS号： 1884712-47-3分子式： C22H22N6O分子量： 386.45描述纯度储存/保存方法别名可溶性/溶解性靶点In vitro(体外研究)
| 产品描述 | |
| 描述 |
CPI-637 is a selective and potent CBP/EP300 bromodomain inhibitor with IC50 values of 0.03 μM, 0.051 μM and 11.0 μM for CBP, EP300 and BRD4 BD-1, respectively, and an EC50 of 0.3 μM for CBP.
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| 纯度 |
≥98%
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| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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| 基本信息 | |
| 别名 |
cpi-637
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| 可溶性/溶解性 |
DMSO : 9.62 mg/mL (24.89 mM; Need ultrasonic)
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| 生物活性 | |
| 靶点 |
BRD4 BD1；CBP；EP300
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| In vitro(体外研究) |
CPI-637 (Compound 28) inhibits MYC expression in AMO-1 cells (EC50 value of 0.60 μM) .
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分子结构图
