NGD 94-1CAS号： 179333-18-7分子式： C18H20N6分子量： 320.39描述应用储存/保存方法形态PK值Ki 数据可溶性/溶解性PubChem CID
| 产品描述 | |
| 描述 |
NGD 94-1 is reported to be a high affinity D4 receptor ligand and is selective over D1, D2, D3 and D5 receptors. In transfected Chinese hamster ovary cells, additionally displays antagonist activity at the human D4.2 receptor. In HEK-293 cells displays agonist activity at the D4.4 receptor.
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| 应用 |
A high affinity D4 receptor ligand that is selective over D1, D2, D3, and D5 receptors
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| 储存/保存方法 |
Store at 4° C
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| 形态 |
Solid
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| 基本信息 | |
| PK值 |
pKa: 12.93 (Predicted), pKb: 6.5 (Predicted)
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| Ki 数据 |
D4.2 receptor: Ki= 3.6 nM (transfected CHO cells)
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| 可溶性/溶解性 |
Soluble in 1eq. HCl (100 mM), and DMSO (100 mM).
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| PubChem CID |
188942
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