Brimonidine

BrimonidineCAS号: 59803-98-4分子式:

C11H10BrN5

分子量: 292.14描述纯度储存/保存方法形态别名外观可溶性/溶解性靶点In vitro(体外研究)

产品描述
描述

Brimonidine (UK 14304) is a full α2-adrenergic receptor (α2-AR) agonist. 

纯度
>98%
储存/保存方法
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
形态
Solid
基本信息
别名
溴莫尼定;UK 14,304;UK 14304;AGN190342
外观
微黄色至黄色结晶性粉末
可溶性/溶解性
DMSO :26 mg/mL (89.0 mM)
生物活性
靶点
α2-adrenergic Receptor.
In vitro(体外研究)
[3H]Brimonidine (UK 14304) is a full agonist at alpha 2-adrenergic receptors. [3H]Brimonidine (UK 14304) labels at least 2 specific binding sites in human brain that both have the characteristics of an alpha 2-adrenergic binding site. GTP decreases agonist binding at both of these sites, but with different potencies at each site.

分子结构图

Brimonidine