SKF 86002 dihydrochlorideCAS号: 116339-68-5分子式: C16H12FN3S.2HCl分子量: 370.27描述纯度储存/保存方法别名外观可溶性/溶解性靶点
产品描述 | |
描述 |
Inhibitor of p38 MAP kinase (IC50 = 0.1 – 1 μM). Potently inhibits LPS-induced IL-1 and TNF-α production in human monocytes (IC50 = 1 μM). Also inhibits 5-lipoxygenase- and cyclooxygenase-mediated arachidonic acid metabolism in RBL-1 cells (IC50 values are 10 and 100 μM respectively). |
纯度 |
98%
|
储存/保存方法 |
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
|
基本信息 | |
别名 |
SKF 86002 2HCl
|
外观 |
powder
|
可溶性/溶解性 |
Soluble to 50 mM in sterile water
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生物活性 | |
靶点 |
p38
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分子结构图