MK-8245 TrifluoroacetateCAS号: 1415559-41-9分子式: C19H17BrF4N6O6分子量: 581.27描述纯度储存/保存方法别名可溶性/溶解性靶点
产品描述 | |
描述 |
MK-8245 trifluoroacetate is a liver-targeting inhibitor of stearoyl-CoA desaturase (SCD) with IC50 of 1 nM for human SCD1 and 3 nM for both rat SCD1 and mouse SCD1, with anti-diabetic and anti-dyslipidemic efficacy. |
纯度 |
>98%
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储存/保存方法 |
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
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基本信息 | |
别名 |
MK 8245 Trifluoroacetate, MK8245 Trifluoroacetate
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可溶性/溶解性 |
10 mM in DMSO
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生物活性 | |
靶点 |
Stearoyl-CoA Desaturase (SCD)
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分子结构图