PD 168077 maleateCAS号： 190383-31-4分子式： C20H22N4O•C4H4O4分子量： 450.49描述应用纯度储存/保存方法形态熔点沸点折射率Ki 数据可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
PD 168077 maleate is a D4DR (D4 dopamine) agonist. >400-fold selectivity over D2 with >300-fold selectivity v.s. D3 subtypes. Generates synaptic translocation of CaMK II to postsynaptic sites in cultured prefrontal cortical neurons.
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| 应用 |
A potent and selective agonist of the dopamine D4 receptor
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| 纯度 |
≥99%
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| 储存/保存方法 |
Desiccate at -20° C
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| 形态 |
Solid
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| 基本信息 | |
| 熔点 |
150-153° C
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| 沸点 |
554.6° C at 760 mmHg (Predicted)
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| 折射率 |
n20D ~1.64 (Predicted)
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| Ki 数据 |
D4 dopamine receptor: Ki= 8.7 nM
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| 可溶性/溶解性 |
Soluble in DMSO (100 mM), and ethanol (25 mM).
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| MDL |
MFCD01321067
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| PubChem CID |
11957665
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