NVP-BHG712 isomer

NVP-BHG712 isomerCAS号: 2245892-85-5分子式: C26H20F3N7O分子量: 503.48描述纯度储存/保存方法可溶性/溶解性靶点In vitro(体外研究)

产品描述
描述
NVP-BHG712 isomer shows conserved non-bonded binding to EPHA2 and EPHB4.
纯度
98%
储存/保存方法
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
基本信息
可溶性/溶解性
H2O:insoluble,DMSO:50 mg/mL (99.31 mM)
生物活性
靶点
EPHA2:163 nM
In vitro(体外研究)
NVP-BHG712 isomer exhibits IC50 of 163 nM and 1660 nM for EPHA2 and EPHA4, respectively[1].